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[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS No. 137565-28-7
[Lys5,MeLeu9,Nle10]-NKA(4-10)( —— )
Catalog No. M22354 CAS No. 137565-28-7
Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 385 | In Stock |
|
| 10MG | 570 | In Stock |
|
| 25MG | 888 | In Stock |
|
| 50MG | 1224 | In Stock |
|
| 100MG | 1647 | In Stock |
|
| 500MG | 3303 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product Name[Lys5,MeLeu9,Nle10]-NKA(4-10)
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NoteResearch use only, not for human use.
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Brief DescriptionHighy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
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DescriptionHighy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetNeurokinin Receptor
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RecptorNK2
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Research Area——
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Indication——
Chemical Information
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CAS Number137565-28-7
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Formula Weight804
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Molecular FormulaC39H65N9O9
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Purity>98% (HPLC)
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Solubilitywater:1 mg/mL
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SMILESCCCC[C@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CNC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](N)CC(O)=O)C(C)C)C(N)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Chassaing et al (1991) Selective agonists of NK-2 binding sites highly active on rat portal vein (NK-3 bioassay). Neuropeptides 19 91 PMID:
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